CBPD-268 [Ligand Id: 13245] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CREB binding lysine acetyltransferase in Human [GtoPdb: 2734] [UniProtKB: Q92793] | ||||||||
| GtoPdb | - | - | 7.96 | pIC50 | 11 | nM | IC50 | J Med Chem (2024) 67: 5275-5304 [PMID:38477974] |
| EP300 lysine acetyltransferase in Human [GtoPdb: 2735] [UniProtKB: Q09472] | ||||||||
| GtoPdb | - | - | 8.02 | pIC50 | 9.5 | nM | IC50 | J Med Chem (2024) 67: 5275-5304 [PMID:38477974] |
| cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2] | ||||||||
| GtoPdb | - | - | 5.74 | pIC50 | 1800 | nM | IC50 | J Med Chem (2024) 67: 5275-5304 [PMID:38477974] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
