GSK682753A [Ligand Id: 13053] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GPR183 in Human [GtoPdb: 81] [UniProtKB: P32249] | ||||||||
| GtoPdb | Determined in a CREB-based reporter assay in HEK293 cells transiently transfected with wild type hGPR183; measuring inhibition of GPR183 constitutive activity. | - | 7.27 | pIC50 | 53.6 | nM | IC50 | J Biol Chem (2011) 286: 29292-29302 [PMID:21673108] |
| GtoPdb | Measuring inhibition of [35S]GTPγS binding to hGPR183 in cell membrane preparations | - | 8.59 | pIC50 | 2.6 | nM | IC50 | J Biol Chem (2011) 286: 29292-29302 [PMID:21673108] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
