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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| NLRP3 in Human [GtoPdb: 1770] [UniProtKB: Q96P20] | ||||||||
| GtoPdb | - | - | 6.99 | pKd | 102.7 | nM | Kd | J Med Chem (2023) 66: 16141-16167 [PMID:38029358] |
| GtoPdb | Inhibition of NLRP3 activation | - | 6.89 | pIC50 | 130 | nM | IC50 | J Med Chem (2023) 66: 16141-16167 [PMID:38029358] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.