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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference | 
|---|---|---|---|---|---|---|---|---|
| ketohexokinase in Human [GtoPdb: 3236] [UniProtKB: P50053] | ||||||||
| GtoPdb | Inhibition of fructose conversion to F1P by KHK in HepG2 liver cells | - | 7.39 | pIC50 | 41 | nM | IC50 | J Med Chem (2023) 66: 15960-15976 [PMID:37992274] | 
| GtoPdb | Biochemical inhibition of hKHK-C and hKHK-A isoforms | - | 7.7 | pIC50 | 20 | nM | IC50 | J Med Chem (2023) 66: 15960-15976 [PMID:37992274] | 
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.