tibremciclib [Ligand Id: 12881] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| cyclin dependent kinase 4 in Human [GtoPdb: 1976] [UniProtKB: P11802] | ||||||||
| GtoPdb | - | - | 8.72 | pIC50 | 1.9 | nM | IC50 | US20210261546A1. Crystal form of compound for inhibiting the activity of cdk4/6 and use thereof (2021) |
| cyclin dependent kinase 6 in Human [GtoPdb: 1978] [UniProtKB: Q00534] | ||||||||
| GtoPdb | - | - | 7.66 | pIC50 | 22 | nM | IC50 | US20210261546A1. Crystal form of compound for inhibiting the activity of cdk4/6 and use thereof (2021) |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
