canlitinib [Ligand Id: 12865] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
Created with Highcharts 10.3.3ValuesChart context menukinase insert domain receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • AXL receptor tyrosine kinase in Human [GtoPdb: 1835] [UniProtKB: P30530]
Created with Highcharts 10.3.3ValuesChart context menuAXL receptor tyrosine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human024681012Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
kinase insert domain receptor in Human [GtoPdb: 1813] [UniProtKB: P35968]
GtoPdb - - 9.42 pIC50 0.38 nM IC50 WO2020216188. Crystal forms of compound, preparation method therefor, pharmaceutical composition and application thereof (2020)
AXL receptor tyrosine kinase in Human [GtoPdb: 1835] [UniProtKB: P30530]
GtoPdb - - 9.62 pIC50 0.24 nM IC50 WO2020216188. Crystal forms of compound, preparation method therefor, pharmaceutical composition and application thereof (2020)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.