PTD10 [Ligand Id: 12687] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187] | ||||||||
| GtoPdb | Inhibition of BTK catalytic activity in a cellular assay | - | 7.01 | pIC50 | 97 | nM | IC50 | Journal of Mediconal Chemistry (2023) : |
| cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2] | ||||||||
| GtoPdb | Measuring target engagement in a NanoBRET competitive displacement assay. | - | 6.97 | pIC50 | 107 | nM | IC50 | Journal of Mediconal Chemistry (2023) : |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
