iodophenpropit [Ligand Id: 1266] activity data from GtoPdb

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  • H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
  • H3 receptor in Rat [GtoPdb: 264] [UniProtKB: Q9QYN8]
Created with Highcharts 10.3.3ValuesChart context menuH3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpKd RatpKi RatpIC50 RatpEC50 Rat0246810Highcharts.com
  • H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
Created with Highcharts 10.3.3ValuesChart context menuH4 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
GtoPdb - - 8.7 pKi 1.99 nM Ki J Pharmacol Exp Ther (2001) 299: 908-14 [PMID:11714875];
Eur J Pharmacol (2002) 453: 33-41 [PMID:12393057]
H3 receptor in Rat [GtoPdb: 264] [UniProtKB: Q9QYN8]
GtoPdb - - 9.1 pKi - - - J Pharmacol Exp Ther (2001) 299: 908-14 [PMID:11714875];
Eur J Pharmacol (2002) 453: 33-41 [PMID:12393057]
H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
GtoPdb - - 7.7 pKi - - - Mol Pharmacol (2001) 59: 434-41 [PMID:11179436]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.