ACT-709478 [Ligand Id: 12647] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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| Cav3.1 in Human [GtoPdb: 535] [UniProtKB: O43497] | ||||||||
| GtoPdb | - | - | 8.19 | pIC50 | 6.4 | nM | IC50 | J Med Chem (2017) 60: 9769-9789 [PMID:29116786] |
| Cav3.2 in Human [GtoPdb: 536] [UniProtKB: O95180] | ||||||||
| GtoPdb | - | - | 7.74 | pIC50 | 18 | nM | IC50 | J Med Chem (2017) 60: 9769-9789 [PMID:29116786] |
| Cav3.3 in Human [GtoPdb: 537] [UniProtKB: Q9P0X4] | ||||||||
| GtoPdb | - | - | 8.12 | pIC50 | 7.5 | nM | IC50 | J Med Chem (2017) 60: 9769-9789 [PMID:29116786] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
