YL5084 [Ligand Id: 12484] activity data from GtoPdb

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  • mitogen-activated protein kinase 8 in Human [GtoPdb: 1496] [UniProtKB: P45983]
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  • mitogen-activated protein kinase 9 in Human [GtoPdb: 1497] [UniProtKB: P45984]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
mitogen-activated protein kinase 8 in Human [GtoPdb: 1496] [UniProtKB: P45983]
GtoPdb - - 5.66 pIC50 2173 nM IC50 J Med Chem (2023) 66: 3356-3371 [PMID:36826833]
mitogen-activated protein kinase 9 in Human [GtoPdb: 1497] [UniProtKB: P45984]
GtoPdb - - 7.15 pIC50 70 nM IC50 J Med Chem (2023) 66: 3356-3371 [PMID:36826833]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.