linzagolix [Ligand Id: 12283] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GnRH1 receptor in Monkey [GtoPdb: 256] | ||||||||
| GtoPdb | Inhibition of GnRH-induced Ca2+ flux in HEK293 cells stably expressing cynomolgus monkey GnRHR | - | 6.35 | pIC50 | 442 | nM | IC50 | Clin Exp Pharmacol Physiol (2022) 49: 1082-1093 [PMID:35690889] |
| GnRH1 receptor in Human [GtoPdb: 256] [UniProtKB: P30968] | ||||||||
| GtoPdb | Inhibition of GnRH-stimulated Ca2+ flux in HEK293 cells stably expressing hGnRHR. | - | 7.44 | pIC50 | 36.7 | nM | IC50 | Clin Exp Pharmacol Physiol (2022) 49: 1082-1093 [PMID:35690889] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
