ACT-660602 [Ligand Id: 12207] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CXCR3 in Human [GtoPdb: 70] [UniProtKB: P49682] | ||||||||
| GtoPdb | Antagonist potency determined by FLIPR calcium mobilization assay, in CHO-K1 cells expressing recombinant CXCR3 receptors with CXCL10 as agonist | - | 8.57 | pIC50 | 2.7 | nM | IC50 | J Med Chem (2022) 65: 11513-11532 [PMID:35947786] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
