TL12-186 [Ligand Id: 12147] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| cereblon in Human [GtoPdb: 3086] [UniProtKB: Q96SW2] | ||||||||
| GtoPdb | Half-maximal inhibitory concentration determined using an AlphaScreen engagement assay, measuring displacement of biotinylated thalidomide from CRBN | - | 7.92 | pIC50 | 12 | nM | IC50 | Cell Chem Biol (2018) 25: 88-99.e6 [PMID:29129717] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
