iclepertin [Ligand Id: 12110] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GlyT1 in Human [GtoPdb: 935] [UniProtKB: P48067] | ||||||||
| GtoPdb | Measuring inhibition of [3H]-glycine uptake in human SK-N-MC cells | - | 8.3 | pIC50 | 5 | nM | IC50 | Clin Transl Sci (2018) 11: 616-623 [PMID:30136756] |
| GlyT1 in Rat [GtoPdb: 935] [UniProtKB: P28572] | ||||||||
| GtoPdb | Inhibition of [3H]-glycine uptake in rat primary neurons | - | 8.28 | pIC50 | 5.2 | nM | IC50 | Clin Transl Sci (2018) 11: 616-623 [PMID:30136756] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
