sulfopin [Ligand Id: 11540] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| peptidylprolyl cis/trans isomerase, NIMA-interacting 1 in Human [GtoPdb: 3171] [UniProtKB: Q13526] | ||||||||
| GtoPdb | Inhibition of Pin1 catalytic activity determined in a chymotrypsin-coupled peptidyl-prolyl isomerization assay (PPIase) assay | - | 6.68 | pKi | 211 | nM | Ki | Nat Chem Biol (2021) 17: 954-963 [PMID:33972797] |
| GtoPdb | Binding to Pin1 in a fluorescence polarization (FP) assay that measured competitive displacement of an N-terminal fluorescein-labeled peptide substrate (Bth-D-pThr-Pip-Nal) | - | 7.77 | pKi | 17 | nM | Ki | Nat Chem Biol (2021) 17: 954-963 [PMID:33972797] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
