NTP42 [Ligand Id: 11537] activity data from GtoPdb

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  • TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
TP receptor in Human [GtoPdb: 346] [UniProtKB: P21731]
GtoPdb Antagonism of U46619-mediated [Ca2+]i mobilization in HEK293 cells expressing TP&aipha; - 7.25 pIC50 56.2 nM IC50 WO2016203314A1. Thromboxane receptor antagonists (2016)
GtoPdb Antagonism of U46619-mediated [Ca2+]i mobilization in HEK293 cells expressing TPβ - 8.08 pIC50 8.25 nM IC50 WO2016203314A1. Thromboxane receptor antagonists (2016)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.