exendin-4 [Ligand Id: 1135] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220] | ||||||||
| GtoPdb | - | - | 9 | pKi | 1 | nM | Ki | Mol Endocrinol (2005) 19: 812-23 [PMID:15528268] |
| GtoPdb | Displacement of GLP-1 from hGLP-1 receptor expressed in CHOK1 cells by exendin-4 | - | 9.18 | pIC50 | 0.66 | nM | IC50 | J Med Chem (2008) 51: 2758-65 [PMID:18412318] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
