EST64454 [Ligand Id: 11343] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • sigma non-opioid intracellular receptor 1 in Human [GtoPdb: 2552] [UniProtKB: Q99720]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
sigma non-opioid intracellular receptor 1 in Human [GtoPdb: 2552] [UniProtKB: Q99720]
GtoPdb Measuring displacement of radiotracer [3H](+)-pentazocine binding to membranes from HEK293 cells expressing human sigma1 receptor. - 7.66 pKi 22 nM Ki J Med Chem (2020) : [PMID:33237785]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.