CpY [Ligand Id: 11314] activity data from GtoPdb

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  • LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
Created with Highcharts 10.3.3ValuesChart context menuLPA1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0]
Created with Highcharts 10.3.3ValuesChart context menuLPA2 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5]
Created with Highcharts 10.3.3ValuesChart context menuLPA3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633]
GtoPdb - - 8.3 pKi 5 nM Ki J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422]
GtoPdb - - 6.3 pEC50 501 nM EC50 J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422]
LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0]
GtoPdb - - 8.7 pKi 2 nM Ki J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422]
GtoPdb - - 7.5 pEC50 31.6 nM EC50 J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422]
LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5]
GtoPdb - - 7.7 pEC50 20 nM EC50 J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.