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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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LPA1 receptor in Human [GtoPdb: 272] [UniProtKB: Q92633] | ||||||||
GtoPdb | - | - | 8.3 | pKi | 5 | nM | Ki | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
GtoPdb | - | - | 6.3 | pEC50 | 501 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
LPA2 receptor in Human [GtoPdb: 273] [UniProtKB: Q9HBW0] | ||||||||
GtoPdb | - | - | 8.7 | pKi | 2 | nM | Ki | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
GtoPdb | - | - | 7.5 | pEC50 | 31.6 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
LPA3 receptor in Human [GtoPdb: 274] [UniProtKB: Q9UBY5] | ||||||||
GtoPdb | - | - | 7.7 | pEC50 | 20 | nM | EC50 | J Pharmacol Exp Ther (2020) 374: 283-294 [PMID:32409422] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.