enerisant [Ligand Id: 11293] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1] | ||||||||
| GtoPdb | Determined using [3H]N-α-methylhistamine binding to the membranes of CHO-K1 cells expressing human recombinant H3 receptors. | - | 8.78 | pKi | 1.65 | nM | Ki | J Pharmacol Exp Ther (2020) 375: 276-285 [PMID:32862143] |
| H3 receptor in Rat [GtoPdb: 264] [UniProtKB: Q9QYN8] | ||||||||
| GtoPdb | - | - | 8.1 | pKi | 7.87 | nM | Ki | J Pharmacol Exp Ther (2020) 375: 276-285 [PMID:32862143] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
