ZYBT1 [Ligand Id: 11193] activity data from GtoPdb

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  • BMX non-receptor tyrosine kinase in Human [GtoPdb: 1942] [UniProtKB: P51813]
Created with Highcharts 10.3.3ValuesChart context menuBMX non-receptor tyrosine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
  • Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
Created with Highcharts 10.3.3ValuesChart context menuBruton tyrosine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • tec protein tyrosine kinase in Human [GtoPdb: 2238] [UniProtKB: P42680]
Created with Highcharts 10.3.3ValuesChart context menutec protein tyrosine kinasepKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BMX non-receptor tyrosine kinase in Human [GtoPdb: 1942] [UniProtKB: P51813]
GtoPdb - - 7.04 pIC50 91 nM IC50 Pharmacol Res Perspect (2020) 8: e00565 [PMID:32790160]
Bruton tyrosine kinase in Human [GtoPdb: 1948] [UniProtKB: Q06187]
GtoPdb - - 7.85 pKi 14 nM Ki Pharmacol Res Perspect (2020) 8: e00565 [PMID:32790160]
GtoPdb - - 9 pIC50 1 nM IC50 Pharmacol Res Perspect (2020) 8: e00565 [PMID:32790160]
tec protein tyrosine kinase in Human [GtoPdb: 2238] [UniProtKB: P42680]
GtoPdb - - 7.6 pIC50 25 nM IC50 Pharmacol Res Perspect (2020) 8: e00565 [PMID:32790160]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.