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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| phosphodiesterase 1C in Human [GtoPdb: 1296] [UniProtKB: Q14123] | ||||||||
| GtoPdb | Biochemical inhibition of recombinant PDE1C catalytic domain (aa147–531). | - | 8.54 | pIC50 | 2.9 | nM | IC50 | J Med Chem (2020) 63: 7867-7879 [PMID:32603117] |
| phosphodiesterase 4D in Human [GtoPdb: 1303] [UniProtKB: Q08499] | ||||||||
| GtoPdb | Biochemical inhibition of recombinant PDE4D2 catalytic domain (aa86–413). | - | 6.16 | pIC50 | 699 | nM | IC50 | J Med Chem (2020) 63: 7867-7879 [PMID:32603117] |
| phosphodiesterase 5A in Human [GtoPdb: 1304] [UniProtKB: O76074] | ||||||||
| GtoPdb | Biochemical inhibition of recombinant PDE5A1 catalytic domain (aa535–860). | - | 6.43 | pIC50 | 370 | nM | IC50 | J Med Chem (2020) 63: 7867-7879 [PMID:32603117] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.