obatoclax [Ligand Id: 11086] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BCL2 apoptosis regulator in Human [GtoPdb: 2844] [UniProtKB: P10415] | ||||||||
| GtoPdb | In vitro antagonism determined in a fluorescence polarisation assay. | - | 5.96 | pKi | 1100 | nM | Ki | Eur J Med Chem (2018) 146: 471-482 [PMID:29407973] |
| Bcl-2-like 1 in Human [GtoPdb: 2845] [UniProtKB: Q07817] | ||||||||
| GtoPdb | In vitro antagonism determined in a fluorescence polarisation assay. | - | 5.33 | pKi | 4690 | nM | Ki | Eur J Med Chem (2018) 146: 471-482 [PMID:29407973] |
| MCL1 apoptosis regulator, BCL2 family member in Human [GtoPdb: 2847] [UniProtKB: Q07820] | ||||||||
| GtoPdb | In vitro antagonism determined in a fluorescence polarisation assay. | - | 5.54 | pKi | 2900 | nM | Ki | Eur J Med Chem (2018) 146: 471-482 [PMID:29407973] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
