adagrasib [Ligand Id: 10888] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • KRAS in Human [GtoPdb: 2824] [UniProtKB: P01116]
Created with Highcharts 10.3.3ValuesChart context menuKRASpKd HumanpKi HumanpIC50 HumanpEC50 Human0123456Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
KRAS in Human [GtoPdb: 2824] [UniProtKB: P01116]
GtoPdb - - 5.43 pKi 3700 nM Ki J Med Chem (2020) null: null [PMID:32250617]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.