GNF4877 [Ligand Id: 10688] activity data from GtoPdb

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  • dual specificity tyrosine phosphorylation regulated kinase 1A in Human [GtoPdb: 2009] [UniProtKB: Q13627]
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  • glycogen synthase kinase 3 beta in Human [GtoPdb: 2030] [UniProtKB: P49841]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
dual specificity tyrosine phosphorylation regulated kinase 1A in Human [GtoPdb: 2009] [UniProtKB: Q13627]
GtoPdb - - 8.22 pIC50 6 nM IC50 Nat Commun (2015) 6: 8372 [PMID:26496802]
glycogen synthase kinase 3 beta in Human [GtoPdb: 2030] [UniProtKB: P49841]
GtoPdb - - 7.8 pIC50 16 nM IC50 Nat Commun (2015) 6: 8372 [PMID:26496802]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.