licogliflozin [Ligand Id: 10654] activity data from GtoPdb

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  • Sodium/glucose cotransporter 1 in Human [GtoPdb: 915] [UniProtKB: P13866]
Created with Highcharts 10.3.3ValuesChart context menuSodium/glucose cotransporter 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
  • Sodium/glucose cotransporter 2 in Human [GtoPdb: 916] [UniProtKB: P31639]
Created with Highcharts 10.3.3ValuesChart context menuSodium/glucose cotransporter 2pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Sodium/glucose cotransporter 1 in Human [GtoPdb: 915] [UniProtKB: P13866]
GtoPdb Measuring inhibition of sodium-dependent [14]C- alpha-methyl-glucopyranoside (AMG) transport into the interior of cells transfected with hSGLT1. - 7.66 pIC50 22 nM IC50 WO2011048112A1. Glycoside derivatives and uses thereof (2011)
Sodium/glucose cotransporter 2 in Human [GtoPdb: 916] [UniProtKB: P31639]
GtoPdb Measuring inhibition of sodium-dependent [14]C- alpha-methyl-glucopyranoside (AMG) transport into the interior of cells transfected with hSGLT2. - 9.3 pIC50 0.5 nM IC50 WO2011048112A1. Glycoside derivatives and uses thereof (2011)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.