compound 16 [PMID: 31977207] [Ligand Id: 10650] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| pyruvate kinase M1/2 in Human [GtoPdb: 3006] [UniProtKB: P14618] | ||||||||
| GtoPdb | Activation of PKM2 kinase activity (promotion of high kinase activity PKM2 tertramer formation) in vitro, by compound 5; described as AC50 in the reference, | - | 7.82 | pEC50 | ~15 | nM | EC50 | J Med Chem (2020) 63: 1597-1611 [PMID:31977207] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
