JNJ-27141491 [Ligand Id: 10586] activity data from GtoPdb

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  • CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
Created with Highcharts 10.3.3ValuesChart context menuCCR2pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597]
GtoPdb Measuring antagonism of 125I-MCP-1binding to human CCR2 expressed by CHO cells in a competition binding assay. - 7.02 pIC50 95 nM IC50 J Pharmacol Exp Ther (2008) 327: 1-9 [PMID:18599682]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.