dTRIM24 [Ligand Id: 10536] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • tripartite motif containing 24 in Human [GtoPdb: 2252] [UniProtKB: O15164]
Created with Highcharts 10.3.3ValuesChart context menutripartite motif containing 24pKd HumanpKi HumanpIC50 HumanpEC50 Human02468Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
tripartite motif containing 24 in Human [GtoPdb: 2252] [UniProtKB: O15164]
GtoPdb Active binding to the TRIM24 bromodomain in TRIM24 ligand-displacement (AlphaScreen) assay. - 6.47 pIC50 337.7 nM IC50 Nat Chem Biol (2018) 14: 405-412 [PMID:29507391]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.