RJW100 [Ligand Id: 10484] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Steroidogenic factor 1 in Human [GtoPdb: 632] [UniProtKB: Q13285] | ||||||||
| GtoPdb | Binding affinity measured using a fluorescence resonance energy transfer (FRET)-based peptide recruitment assay. | - | 7.5 | pEC50 | 31.6 | nM | EC50 | J Med Chem (2011) 54: 2266-81 [PMID:21391689] |
| Liver receptor homolog-1 in Human [GtoPdb: 633] [UniProtKB: O00482] | ||||||||
| GtoPdb | Measuring LRH-1-mediated transcriptional activation in a luciferase reporter assay. | - | 5.82 | pEC50 | 1500 | nM | EC50 | J Med Chem (2019) 62: 11022-11034 [PMID:31419141] |
| GtoPdb | Binding affinity measured using a fluorescence resonance energy transfer (FRET)-based peptide recruitment assay. | - | 6.6 | pEC50 | 251 | nM | EC50 | J Med Chem (2011) 54: 2266-81 [PMID:21391689] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
