compound 16 [PMID: 31498617] [Ligand Id: 10482] activity data from GtoPdb
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| MRGPRX1 in Human [GtoPdb: 156] [UniProtKB: Q96LB2] | ||||||||
| GtoPdb | Agonist activity at human MRGPRX1 stably expressed in HEK293 cells by FLIPR claciun mobilisation assay. | - | 7.3 | pEC50 | 50 | nM | EC50 | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
| δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143] | ||||||||
| GtoPdb | Receptor binding in a radioligand displacement assay using [3H]DADLE as tracer. | - | 5.61 | pKi | 2470 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
| κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145] | ||||||||
| GtoPdb | Receptor binding in a radioligand displacement assay using [3H]U-69,593 as tracer. | - | 4.92 | pKi | 12100 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
| μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
| GtoPdb | Receptor binding in a radioligand displacement assay using [3H]DAMGO as tracer. | - | 5.43 | pKi | 3730 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
