Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
MRGPRX1 in Human [GtoPdb: 156] [UniProtKB: Q96LB2] | ||||||||
GtoPdb | Agonist activity at human MRGPRX1 stably expressed in HEK293 cells by FLIPR claciun mobilisation assay. | - | 7.3 | pEC50 | 50 | nM | EC50 | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143] | ||||||||
GtoPdb | Receptor binding in a radioligand displacement assay using [3H]DADLE as tracer. | - | 5.61 | pKi | 2470 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145] | ||||||||
GtoPdb | Receptor binding in a radioligand displacement assay using [3H]U-69,593 as tracer. | - | 4.92 | pKi | 12100 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372] | ||||||||
GtoPdb | Receptor binding in a radioligand displacement assay using [3H]DAMGO as tracer. | - | 5.43 | pKi | 3730 | nM | Ki | J Med Chem (2019) 62: 8631-8641 [PMID:31498617] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.