compound E22 [PMID: 31298542] [Ligand Id: 10437] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| AKT serine/threonine kinase 1 in Human [GtoPdb: 1479] [UniProtKB: P31749] | ||||||||
| GtoPdb | - | - | 8.86 | pIC50 | 1.37 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| AKT serine/threonine kinase 2 in Human [GtoPdb: 1480] [UniProtKB: P31751] | ||||||||
| GtoPdb | - | - | 8.92 | pIC50 | 1.2 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| Rho associated coiled-coil containing protein kinase 1 in Human [GtoPdb: 1503] [UniProtKB: Q13464] | ||||||||
| GtoPdb | - | - | 7.19 | pIC50 | 64 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| ribosomal protein S6 kinase B1 in Human [GtoPdb: 1525] [UniProtKB: P23443] | ||||||||
| GtoPdb | - | - | 8.05 | pIC50 | 8.9 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| ribosomal protein S6 kinase A1 in Human [GtoPdb: 1527] [UniProtKB: Q15418] | ||||||||
| GtoPdb | - | - | 6.88 | pIC50 | 131 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| protein kinase A in Human [GtoPdb: 1694] | ||||||||
| GtoPdb | - | - | 9.52 | pIC50 | 0.3 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
| AKT serine/threonine kinase 3 in Human [GtoPdb: 2286] [UniProtKB: Q9Y243] | ||||||||
| GtoPdb | - | - | 8.77 | pIC50 | 1.7 | nM | IC50 | J Med Chem (2019) 62: 7264-7288 [PMID:31298542] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
