zetomipzomib [Ligand Id: 10409] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| proteasome 20S subunit beta 2 in Human [GtoPdb: 2405] [UniProtKB: P49721] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in MOLT-4 (human T cell leukemia) cell lysate using the ProCISE ELISA. | - | 6.22 | pIC50 | 604 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
| proteasome 20S subunit beta 5 in Human [GtoPdb: 2406] [UniProtKB: P28074] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in MOLT-4 (human T cell leukemia) cell lysate using the ProCISE ELISA. | - | 6.16 | pIC50 | 688 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
| proteasome 20S subunit beta 8 in Human [GtoPdb: 2408] [UniProtKB: P28062] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in MOLT-4 (human T cell leukemia) cells using the ProCISE ELISA. | - | 7.41 | pIC50 | 39 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
| proteasome 20S subunit beta 8 in Mouse [GtoPdb: 2408] [UniProtKB: P28063] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in A20 (mouse B-cell lymphoma) cell lysate using the ProCISE ELISA. | - | 7.24 | pIC50 | 57 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
| proteasome 20S subunit beta 9 in Human [GtoPdb: 2409] [UniProtKB: P28065] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in MOLT-4 (human T cell leukemia) cell lysate using the ProCISE ELISA. | - | 6.88 | pIC50 | 131 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
| proteasome 20S subunit beta 9 in Mouse [GtoPdb: 2409] [UniProtKB: P28076] | ||||||||
| GtoPdb | Inhibition of proteolytic activity measured in A20 (mouse B-cell lymphoma) cell lysate using the ProCISE ELISA. | - | 6.75 | pIC50 | 179 | nM | IC50 | J Med Chem (2018) 61: 11127-11143 [PMID:30380863] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
