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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
mitogen-activated protein kinase 8 in Human [GtoPdb: 1496] [UniProtKB: P45983] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 7.49 | pIC50 | 32 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
mitogen-activated protein kinase 9 in Human [GtoPdb: 1497] [UniProtKB: P45984] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 7.23 | pIC50 | 59 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
mitogen-activated protein kinase 10 in Human [GtoPdb: 1498] [UniProtKB: P53779] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 6.97 | pIC50 | 107 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
leukocyte receptor tyrosine kinase in Human [GtoPdb: 1838] [UniProtKB: P29376] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 6.25 | pKi | 567 | nM | Ki | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
CDC like kinase 2 in Human [GtoPdb: 1991] [UniProtKB: P49760] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 6.58 | pIC50 | 261 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
dual specificity tyrosine phosphorylation regulated kinase 3 in Human [GtoPdb: 2012] [UniProtKB: O43781] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 6.98 | pIC50 | 104 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
leucine rich repeat kinase 2 in Human [GtoPdb: 2059] [UniProtKB: Q5S007] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 9 | pIC50 | 1 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
testis specific serine kinase 1B in Human [GtoPdb: 2257] [UniProtKB: Q9BXA7] | ||||||||
GtoPdb | Measuring in vitro enzyme inhibitory activity. | - | 6.66 | pIC50 | 217 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
TTK protein kinase in Human [GtoPdb: 2264] [UniProtKB: P33981] | ||||||||
GtoPdb | In vitro inhibitory activity using the proprietary LanthaScreen Eu kinase binding assay. | - | 9.15 | pIC50 | 0.7 | nM | IC50 | J Med Chem (2019) 62: 4401-4410 [PMID:30998356] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.