stanozolol [Ligand Id: 10369] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2079587
  • Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
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  • Androgen receptor in Rat [GtoPdb: 628] [UniProtKB: P15207]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
GtoPdb Measured in a DrugMatrix estrogen receptor α radioligand binding assay using [3H] estradiol as tracer. - 6.95 pIC50 113 nM IC50 DrugMatrix in vitro pharmacology data. National Toxicology Program
Androgen receptor in Rat [GtoPdb: 628] [UniProtKB: P15207]
GtoPdb Measured in a DrugMatrix in vitro androgen receptor radioligand binding assay using [3H] mibolerone as tracer. - 7.66 pIC50 22 nM IC50 DrugMatrix in vitro pharmacology data. National Toxicology Program

ChEMBL data shown on this page come from version 35:

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]