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ChEMBL ligand: CHEMBL2079587 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372] | ||||||||
GtoPdb | Measured in a DrugMatrix estrogen receptor α radioligand binding assay using [3H] estradiol as tracer. | - | 6.95 | pIC50 | 113 | nM | IC50 | DrugMatrix in vitro pharmacology data. National Toxicology Program |
Androgen receptor in Rat [GtoPdb: 628] [UniProtKB: P15207] | ||||||||
GtoPdb | Measured in a DrugMatrix in vitro androgen receptor radioligand binding assay using [3H] mibolerone as tracer. | - | 7.66 | pIC50 | 22 | nM | IC50 | DrugMatrix in vitro pharmacology data. National Toxicology Program |
ChEMBL data shown on this page come from version 35:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]