Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
K2P2.1 in Human [GtoPdb: 514] [UniProtKB: O95069] | ||||||||
GtoPdb | Measuring GI‐530139-induced enhanced current via single hTREK1 channels measured at +60 mV in the inside‐out manual patch configuration, in a concentration–response experiment. | - | 6.05 | pEC50 | 890 | nM | EC50 | Br J Pharmacol (2018) 175: 2272-2283 [PMID:29150838] |
GtoPdb | Measuring 86Rb efflux by TREK1 induced by GI‐530159 at 70 mM potassium. | - | 6.12 | pEC50 | 760 | nM | EC50 | Br J Pharmacol (2018) 175: 2272-2283 [PMID:29150838] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.