Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
diacylglycerol lipase α in Human [GtoPdb: 1396] [UniProtKB: Q9Y4D2] | ||||||||
GtoPdb | - | - | 7.89 | pIC50 | 13 | nM | IC50 | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
GtoPdb | Inhibition of recombinant human DAGα in a biochemical assay with para-nitrophenylbutyrate as a surrogate substrate. | - | 8.5 | pIC50 | - | - | - | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
diacylglycerol lipase β in Human [GtoPdb: 1397] [UniProtKB: Q8NCG7] | ||||||||
GtoPdb | Inhibition of recombinant human DAGβ in a biochemical assay with para-nitrophenylbutyrate as a surrogate substrate. | - | 8.1 | pIC50 | - | - | - | J Am Chem Soc (2015) 137: 8851-7 [PMID:26083464] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.