NPC 18565   Click here for help

GtoPdb Ligand ID: 658

Synonyms: [D-Arg(Hyp3,D-Hyp7(transpropyl),Oic8)des-Arg9]bradykinin | des-Arg9 fragment of NPC 17731 | NPC-18565 | NPC18565
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Selectivity at GPCRs
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Target Sp. Type Action Value Parameter Concentration range (M) Reference
B1 receptor Hs Antagonist Antagonist 10.2 pKi - 1
pKi 10.2 [1]
B2 receptor Hs Antagonist Antagonist 6.6 pKi - 1
pKi 6.6 [1]