[125I]iodovinyl-TBZ   Click here for help

GtoPdb Ligand ID: 4764

Synonyms: [125I]-iodovinyl-TBZ  | [125I]-iodovinyltetrabenazine
 Ligand is labelled  Ligand is radioactive
Compound class: Synthetic organic
Comment: The structure of the ligand is not specified in the available literature. Our ligand page for tetrabenazine shows the structure of the un-labelled analogue.
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Ligand Activity Visualisation Charts

These are box plot that provide a unique visualisation, summarising all the activity data for a ligand taken from ChEMBL and GtoPdb across multiple targets and species. Click on a plot to see the median, interquartile range, low and high data points. A value of zero indicates that no data are available. A separate chart is created for each target, and where possible the algorithm tries to merge ChEMBL and GtoPdb targets by matching them on name and UniProt accession, for each available species. However, please note that inconsistency in naming of targets may lead to data for the same target being reported across multiple charts.

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View interactive charts of activity data across species
Selectivity at transporters
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
Vesicular monoamine transporter 2 Hs Inhibitor Inhibition 8.1 pKd - 1
⤷ pKd 8.1 (Kd 8.2x10-9 M) [1]