[125I]HPP-HOE140   Click here for help

GtoPdb Ligand ID: 11436

Synonyms: [125I]-3-4-hydroxyphenyl-propionyl-d-Arg0-[Hyp3,Thi5,d-Tic7,Oic8]bradykinin [2]
 Ligand is labelled  Ligand is radioactive
Compound class: Peptide or derivative
Comment: This is a radio-labelled antagonist probe for B2 receptors [1-3]. It is a derivative of icatibant (HOE140).
Selectivity at GPCRs
Key to terms and symbols Click column headers to sort
Target Sp. Type Action Value Parameter Concentration range (M) Reference
B2 receptor Hs Antagonist Antagonist - - - 1,3
⤷ [1,3]