PF-06751979 [Ligand Id: 9943] activity data from GtoPdb

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  • beta-secretase 1 in Human [GtoPdb: 2330] [UniProtKB: P56817]
Created with Highcharts 10.3.3ValuesChart context menubeta-secretase 1pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
beta-secretase 1 in Human [GtoPdb: 2330] [UniProtKB: P56817]
GtoPdb - - 8.14 pIC50 7.3 nM IC50 J Med Chem (2018) 61: 4476-4504 [PMID:29613789]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.