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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
activin A receptor type IL in Human [GtoPdb: 1784] [UniProtKB: P37023] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 7.33 | pIC50 | 47 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
mechanistic target of rapamycin kinase in Human [GtoPdb: 2109] [UniProtKB: P42345] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 8.36 | pIC50 | 4.4 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit alpha in Human [GtoPdb: 2153] [UniProtKB: P42336] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 8.66 | pIC50 | 2.2 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit beta in Human [GtoPdb: 2154] [UniProtKB: P42338] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 6.75 | pIC50 | 176 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit delta in Human [GtoPdb: 2155] [UniProtKB: O00329] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 8.4 | pIC50 | 4 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
phosphatidylinositol-4,5-bisphosphate 3-kinase catalytic subunit gamma in Human [GtoPdb: 2156] [UniProtKB: P48736] | ||||||||
GtoPdb | Using a radiometric protein kinase (33PanQinase activity) assay. | - | 6.69 | pIC50 | 203 | nM | IC50 | Mol Cancer Ther (2015) 14: 1095-106 [PMID:25700704] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.