BRD3444 [Ligand Id: 9648] activity data from GtoPdb and ChEMBL
Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
| ChEMBL ligand: CHEMBL3560390 |
|---|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Plasmodium falciparum phenylalanine--tRNA ligase alpha subunit in Plasmodium falciparum 3D7 [GtoPdb: 2954] [UniProtKB: Q8I246] | ||||||||
| GtoPdb | - | - | 7.34 | pIC50 | 46 | nM | IC50 | Nature (2016) 538: 344-349 [PMID:27602946] |
| GtoPdb | Parasite late stage (IV–V) gametocyte assay | - | 6.18 | pEC50 | 663 | nM | EC50 | Nature (2016) 538: 344-349 [PMID:27602946] |
| Plasmodium falciparum phenylalanine--tRNA ligase alpha subunit in Plasmodium falciparum Dd2 [GtoPdb: 2954] | ||||||||
| GtoPdb | Parasite growth inhibition assay | - | 8.05 | pEC50 | 9 | nM | EC50 | Nature (2016) 538: 344-349 [PMID:27602946] |
ChEMBL data shown on this page come from version 28:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]
This work is licensed under a Creative Commons Attribution-ShareAlike 4.0 International License