SPM-354 [Ligand Id: 9493] activity data from GtoPdb

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  • S1P1 receptor in Human [GtoPdb: 275] [UniProtKB: P21453]
Created with Highcharts 10.3.3ValuesChart context menuS1P1 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpA2 Human0246810Highcharts.com
  • S1P3 receptor in Human [GtoPdb: 277] [UniProtKB: Q99500]
Created with Highcharts 10.3.3ValuesChart context menuS1P3 receptorpKd HumanpKi HumanpIC50 HumanpEC50 HumanpA2 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
S1P1 receptor in Human [GtoPdb: 275] [UniProtKB: P21453]
GtoPdb In a β-arrestin assay. - 7.85 pA2 - - - Mol Pharmacol (2016) 89: 176-86 [PMID:26494861]
S1P3 receptor in Human [GtoPdb: 277] [UniProtKB: Q99500]
GtoPdb In a β-arrestin assay. - 9.3 pA2 - - - Mol Pharmacol (2016) 89: 176-86 [PMID:26494861]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.