human GIP(3-42)NH2 [Ligand Id: 8970] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| GIP receptor in Human [GtoPdb: 248] [UniProtKB: P48546] | ||||||||
| GtoPdb | Measuring in vitro inhibition of native GIP-induced cAMP accumulation at [GIP] of 10 pM and 1 nM. | - | 7.04 | pIC50 | 92 | nM | IC50 | Am J Physiol Endocrinol Metab (2006) 291: E468-75 [PMID:16608883] |
| GtoPdb | Binding affinity for the human receptor expressed in COS7 cells. | - | 7.66 | pIC50 | 22 | nM | IC50 | Am J Physiol Endocrinol Metab (2006) 291: E468-75 [PMID:16608883] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
