ensartinib [Ligand Id: 8959] activity data from GtoPdb

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  • MET proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1815] [UniProtKB: P08581]
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  • ALK receptor tyrosine kinase in Human [GtoPdb: 1839] [UniProtKB: Q9UM73]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
MET proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1815] [UniProtKB: P08581]
GtoPdb Result from DiscoveRx KINOMEscan® selectivity screen. - 9.13 pIC50 0.74 nM IC50 Cancer Res (2011) 71: 4920-31 [PMID:21613408]
ALK receptor tyrosine kinase in Human [GtoPdb: 1839] [UniProtKB: Q9UM73]
GtoPdb Result from DiscoveRx KINOMEscan® selectivity screen. - 9.4 pIC50 <0.4 nM IC50 Cancer Res (2011) 71: 4920-31 [PMID:21613408]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.