compound 7 [WO2012007375] [Ligand Id: 8085] activity data from GtoPdb

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  • interleukin 1 receptor associated kinase 1 in Human [GtoPdb: 2042] [UniProtKB: P51617]
Created with Highcharts 10.3.3ValuesChart context menuinterleukin 1 receptor associated kinase 1pKd HumanpKi HumanpIC50 HumanpEC50 Human01234567Highcharts.com
  • interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3]
Created with Highcharts 10.3.3ValuesChart context menuinterleukin 1 receptor associated kinase 4pKd HumanpKi HumanpIC50 HumanpEC50 Human0246810Highcharts.com
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
interleukin 1 receptor associated kinase 1 in Human [GtoPdb: 2042] [UniProtKB: P51617]
GtoPdb - - 6.01 pIC50 983 nM IC50 WO2012007375. Pyrazolo [1, 5a] pyrimidine and thieno [3, 2b] pyrimidine derivatives as irak4 modulators. (2012)
interleukin 1 receptor associated kinase 4 in Human [GtoPdb: 2045] [UniProtKB: Q9NWZ3]
GtoPdb - - 8.1 pIC50 8 nM IC50 WO2012007375. Pyrazolo [1, 5a] pyrimidine and thieno [3, 2b] pyrimidine derivatives as irak4 modulators. (2012)

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.