cephalexin [Ligand Id: 4832] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1727 (Alsporin, Anhydrous cephalexin, Carnosporin, Cefadros, Cefaleksin, Cefalexin, Cefalexina, Cefalexin anhydrous, Cefalexine, Cephalexin anhydrous, Cephamasten, Durantel, Efalexin, Felexin, Garasin, Iwalexin, Keflet, Keflex, Kefloridina, Keftab, Lilly-66873, Mamalexin, NSC-758162, Oracocin, Pyassan, S-6437, Sinthecillin, Taicelexin, Uphalexin) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| Peptide transporter 2/Oligopeptide transporter, kidney isoform in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3325] [GtoPdb: 985] [UniProtKB: Q63424] | ||||||||
| ChEMBL | TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in SKPT cells | F | 4.12 | pKi | 75000 | nM | Ki | Eur J Pharm Biopharm (2005) 59: 17-24 [PMID:15567297] |
| ChEMBL | TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing LLC-PK1 cells | F | 4.31 | pKi | 49000 | nM | Ki | Am J Physiol (1997) 273: F706-F711 [PMID:9374833] |
| Peptide transporter 2/Solute carrier family 15 member 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1743125] [GtoPdb: 985] [UniProtKB: Q16348] | ||||||||
| ChEMBL | TP_TRANSPORTER: inhibition of Gly-Sar uptake in SKPT cells | F | 4.17 | pKi | 68200 | nM | Ki | J Biol Chem (1995) 270: 25672-25677 [PMID:7592745] |
ChEMBL data shown on this page come from version 34:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
