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ChEMBL ligand: CHEMBL258764 |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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5-HT3A in Human [GtoPdb: 379] | ||||||||
GtoPdb | - | - | 4.93 | pIC50 | 11760 | nM | IC50 | J Pharmacol Exp Ther (1999) 290: 129-35 [PMID:10381768] |
5-HT3A in Mouse [GtoPdb: 379] | ||||||||
GtoPdb | - | - | 5.35 | pIC50 | 4500 | nM | IC50 |
J Pharmacol Exp Ther (1999) 290: 129-35 [PMID:10381768]; Biol Pharm Bull (2009) 32: 861-7 [PMID:19420755] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]