Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
CatSper1 in Mouse [GtoPdb: 388] [UniProtKB: Q91ZR5] | ||||||||
GtoPdb | Whole cell patch clamp | - | 5 | pIC50 | 10000 | nM | IC50 | Nature (2006) 439: 737-40 [PMID:16467839] |
CatSper2 in Mouse [GtoPdb: 389] [UniProtKB: A2ARP9] | ||||||||
GtoPdb | Whole cell patch clamp. | - | 5 | pIC50 | 10000 | nM | IC50 | Mol Hum Reprod (2011) 17: 478-99 [PMID:21642646] |
CatSper3 in Mouse [GtoPdb: 390] [UniProtKB: Q80W99] | ||||||||
GtoPdb | Whole cell patch clamp electrophysiology. | - | 5 | pIC50 | 10000 | nM | IC50 | Nature (2006) 439: 737-40 [PMID:16467839] |
CatSper4 in Mouse [GtoPdb: 391] [UniProtKB: Q8BVN3] | ||||||||
GtoPdb | Whole cell patch clamp electrophysiology. | - | 5 | pIC50 | 10000 | nM | IC50 | Nature (2006) 439: 737-40 [PMID:16467839] |
TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8] | ||||||||
GtoPdb | - | - | 5.5 | pIC50 | 3550 | nM | IC50 | J Neurosci (2005) 25: 4052-61 [PMID:15843607] |
TRPM6 in Human [GtoPdb: 498] [UniProtKB: Q9BX84] | ||||||||
GtoPdb | - | - | 7 | pIC50 | 100 | nM | IC50 | |
TRPV1 in Human [GtoPdb: 507] [UniProtKB: Q8NER1] | ||||||||
GtoPdb | - | - | 7 | pIC50 | 90 | nM | IC50 | |
GtoPdb | - | - | 7 | pIC50 | - | - | - | Br J Pharmacol (2001) 132: 1084-94 [PMID:11226139] |
TRPV1 in Rat [GtoPdb: 507] [UniProtKB: O35433] | ||||||||
GtoPdb | - | - | 6.7 | pIC50 | - | - | - | Br J Pharmacol (2001) 132: 1084-94 [PMID:11226139] |
TRPV2 in Human [GtoPdb: 508] [UniProtKB: Q9Y5S1] | ||||||||
GtoPdb | - | - | 6.2 | pIC50 | 600 | nM | IC50 | |
TRPV2 in Mouse [GtoPdb: 508] [UniProtKB: Q9WTR1] | ||||||||
GtoPdb | - | - | 6.2 | pIC50 | - | - | - | Nature (1999) 398: 436-41 [PMID:10201375] |
TRPV3 in Mouse [GtoPdb: 509] [UniProtKB: Q8K424] | ||||||||
GtoPdb | Patch clamp electrophysiology | - | 6 | pIC50 | - | - | - | Science (2002) 296: 2046-9 [PMID:12016205] |
TRPV4 in Rat [GtoPdb: 510] [UniProtKB: Q9ERZ8] | ||||||||
GtoPdb | - | - | 6.7 | pIC50 | - | - | - | J Neurosci (2002) 22: 6408-14 [PMID:12151520] |
TRPV5 in Human [GtoPdb: 511] [UniProtKB: Q9NQA5] | ||||||||
GtoPdb | - | - | 6.9 | pIC50 | 121 | nM | IC50 | |
TRPV5 in Rabbit [GtoPdb: 511] | ||||||||
GtoPdb | - | - | 6.95 | pIC50 | 111 | nM | IC50 | Br J Pharmacol (2001) 134: 453-62 [PMID:11588099] |
TRPV6 in Mouse [GtoPdb: 512] [UniProtKB: Q91WD2] | ||||||||
GtoPdb | - | - | 5 | pIC50 | 9000 | nM | IC50 | J Physiol (Lond.) (2001) 537: 747-61 [PMID:11744752] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.